WO2009068275A3 - α-AMINOSÄUREDERIVATE ZUR LÖSLICHKEITSVERBESSERUNG - Google Patents
α-AMINOSÄUREDERIVATE ZUR LÖSLICHKEITSVERBESSERUNG Download PDFInfo
- Publication number
- WO2009068275A3 WO2009068275A3 PCT/EP2008/010045 EP2008010045W WO2009068275A3 WO 2009068275 A3 WO2009068275 A3 WO 2009068275A3 EP 2008010045 W EP2008010045 W EP 2008010045W WO 2009068275 A3 WO2009068275 A3 WO 2009068275A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- amino acid
- acid derivatives
- improving solubility
- solubility
- improving
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4973—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom
- A61K8/498—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom having 6-membered rings or their condensed derivatives, e.g. coumarin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
- A61K8/0216—Solid or semisolid forms
- A61K8/022—Powders; Compacted Powders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/36—Carboxylic acids; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
- A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/4946—Imidazoles or their condensed derivatives, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/4953—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom containing pyrimidine ring derivatives, e.g. minoxidil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
- A61K2800/26—Optical properties
- A61K2800/262—Transparent; Translucent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
- A61K2800/30—Characterized by the absence of a particular group of ingredients
- A61K2800/31—Anhydrous
Abstract
Die Erfindung betrifft die Verwendung von α-Aminosäurederivaten zur Löslichkeitsverbesserung von schwerlöslichen Substanzen in Wasser oder wässrigen Lösungen, sowie Mischungen und bevorzugte Zubereitungen.
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2010535285A JP2011504891A (ja) | 2007-11-29 | 2008-11-27 | 溶解性を改良するためのα−アミノ酸誘導体 |
US12/745,143 US8293784B2 (en) | 2007-11-29 | 2008-11-27 | α-amino acid derivatives for improving solubility |
EP08853958A EP2211827A2 (de) | 2007-11-29 | 2008-11-27 | Alpha-aminosäurederivate zur löslichkeitsverbesserung |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102007057543.4 | 2007-11-29 | ||
DE102007057543A DE102007057543A1 (de) | 2007-11-29 | 2007-11-29 | a-Aminosäurederivate zur Löslichkeitsverbesserung |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2009068275A2 WO2009068275A2 (de) | 2009-06-04 |
WO2009068275A3 true WO2009068275A3 (de) | 2010-09-23 |
Family
ID=40377294
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP2008/010045 WO2009068275A2 (de) | 2007-11-29 | 2008-11-27 | α-AMINOSÄUREDERIVATE ZUR LÖSLICHKEITSVERBESSERUNG |
Country Status (5)
Country | Link |
---|---|
US (1) | US8293784B2 (de) |
EP (1) | EP2211827A2 (de) |
JP (1) | JP2011504891A (de) |
DE (1) | DE102007057543A1 (de) |
WO (1) | WO2009068275A2 (de) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP6295261B2 (ja) * | 2012-10-12 | 2018-03-14 | ロレアル | 少なくとも一種のヒドロトロープ及び少なくとも一種の活性化合物を含む化粧品組成物 |
CN105963244A (zh) * | 2016-01-15 | 2016-09-28 | 赵鸣 | 注射用青蒿琥酯制剂及其应用 |
JP7194517B2 (ja) * | 2017-05-30 | 2022-12-22 | 花王株式会社 | 皮膚化粧料 |
CN110785161B (zh) | 2017-06-23 | 2023-06-20 | 宝洁公司 | 用于改善皮肤外观的组合物和方法 |
KR20210011964A (ko) | 2018-07-03 | 2021-02-02 | 더 프록터 앤드 갬블 캄파니 | 피부 병태를 치료하는 방법 |
US10959933B1 (en) | 2020-06-01 | 2021-03-30 | The Procter & Gamble Company | Low pH skin care composition and methods of using the same |
JP2023528616A (ja) | 2020-06-01 | 2023-07-05 | ザ プロクター アンド ギャンブル カンパニー | ビタミンb3化合物の皮膚への浸透を改善する方法 |
Citations (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4980165A (en) * | 1989-01-27 | 1990-12-25 | Genetics Institute, Inc. | Pharmaceutical formulations of plasminogen activator proteins |
CH685561A5 (de) * | 1992-01-27 | 1995-08-15 | Polygon Chemie Ag | Verwendung von von beta-Alanin und dessen Homologen abgeleiteten Tensiden zur Verbesserung der Wasserlöslichkeit von Farbstoffen und optischen Aufhellern. |
US20030114324A1 (en) * | 2001-12-14 | 2003-06-19 | Rainer Lange | Cleansing compositions and their use in feminine hygiene wipes |
US20040043940A1 (en) * | 2000-03-24 | 2004-03-04 | Buenger Joachim | Use of ectoin or ectoin derivatives for protecting stress proteins in the skin |
EP1407758A1 (de) * | 2002-10-10 | 2004-04-14 | Beiersdorf AG | Fettfreie Sonnenschutzmittel |
US20060029563A1 (en) * | 2002-12-30 | 2006-02-09 | Jean-Noel Thorel | Cutanceous metabolic bio-activator |
US20070027223A1 (en) * | 2005-07-28 | 2007-02-01 | Werner Bruchert | Foamed preparation |
US20070155695A1 (en) * | 2004-01-19 | 2007-07-05 | Corinna Wirth | Flavonoid complexes with cyclodextrins |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4116123B4 (de) | 1991-05-17 | 2006-03-09 | Merck Patent Gmbh | Mittel zur Behandlung von Hauterkrankungen |
JPH05301813A (ja) * | 1991-10-15 | 1993-11-16 | Kao Corp | 皮膚外用剤 |
DE4308282C2 (de) | 1993-03-16 | 1994-12-22 | Beiersdorf Ag | Vorzugsweise in Form von Mikrosphärulen vorliegende galenische Matrices |
FR2755856B1 (fr) | 1996-11-21 | 1999-01-29 | Merck Clevenot Laboratoires | Microcapsules de chitine ou de derives de chitine contenant une substance hydrophobe, notamment un filtre solaire et procede de preparation de telles microcapsules |
CN1293565A (zh) * | 1998-03-16 | 2001-05-02 | 宝洁公司 | 调节皮肤外观的组合物 |
ATE546131T1 (de) | 1998-08-13 | 2012-03-15 | Sol Gel Technologies Ltd | Verfahren zur herstellung von mit funktionalisierten molekülen beladene oxid- mikrokapseln und die daraus erhaltenen produkte |
US6238650B1 (en) | 1999-05-26 | 2001-05-29 | Sol-Gel Technologies Ltd. | Sunscreen composition containing sol-gel microcapsules |
US6436375B1 (en) | 1999-05-25 | 2002-08-20 | Sol-Gel Technologies Ltd. | Method for obtaining photostable sunscreen compositions |
DE60231272D1 (de) * | 2001-06-26 | 2009-04-09 | Oreal | Zusammensetzungen, die eine wenig lösliche Verbindung und ein lipophiles Aminosäurederivat enthalten, und entsprechende Verwendungen und Verfahren |
DE10133202A1 (de) | 2001-07-07 | 2003-01-16 | Beiersdorf Ag | Osmolyte enthaltende kosmetische und dermatologische Zubereitungen zur Behandlung und aktiven Prävention trockener Haut und anderer negativer Veränderungen der physiologischen Homöostase der gesunden Haut |
DE10232595A1 (de) | 2002-07-18 | 2004-02-05 | Merck Patent Gmbh | Lichtschutzmittel |
DE10240923A1 (de) * | 2002-09-02 | 2004-03-04 | Merck Patent Gmbh | Flavonoid-Derivate zur Ekzem-Behandlung |
DE10244282A1 (de) | 2002-09-23 | 2004-04-01 | Merck Patent Gmbh | Zubereitung mit antioxidanten Eigenschaften |
DE10316666B4 (de) * | 2003-04-10 | 2015-04-09 | Beiersdorf Ag | Kosmetische oder dermatologische Zubereitungen mit einer Kombination von Kreatinin mit Kreatin und Coenzym Q10 |
JP5241054B2 (ja) * | 2004-02-27 | 2013-07-17 | ロート製薬株式会社 | コラーゲン合成促進用組成物 |
JP2005298452A (ja) * | 2004-04-16 | 2005-10-27 | Saga Seiyaku Kk | アズレン誘導体含有の水性液剤の安定化法 |
JP3878629B2 (ja) * | 2004-08-04 | 2007-02-07 | ピアス株式会社 | 複合化水性ゲルとその製造方法、並びに、その複合化水性ゲルを含有するゲル化製剤、皮膚外用剤、及び化粧料 |
DE102006037724A1 (de) | 2006-08-11 | 2008-02-14 | Merck Patent Gmbh | Verwendung von Ascorbinsäurederivaten zur Funktionalisierung von Matrices |
-
2007
- 2007-11-29 DE DE102007057543A patent/DE102007057543A1/de not_active Withdrawn
-
2008
- 2008-11-27 WO PCT/EP2008/010045 patent/WO2009068275A2/de active Application Filing
- 2008-11-27 JP JP2010535285A patent/JP2011504891A/ja active Pending
- 2008-11-27 EP EP08853958A patent/EP2211827A2/de not_active Withdrawn
- 2008-11-27 US US12/745,143 patent/US8293784B2/en not_active Expired - Fee Related
Patent Citations (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4980165A (en) * | 1989-01-27 | 1990-12-25 | Genetics Institute, Inc. | Pharmaceutical formulations of plasminogen activator proteins |
CH685561A5 (de) * | 1992-01-27 | 1995-08-15 | Polygon Chemie Ag | Verwendung von von beta-Alanin und dessen Homologen abgeleiteten Tensiden zur Verbesserung der Wasserlöslichkeit von Farbstoffen und optischen Aufhellern. |
US20040043940A1 (en) * | 2000-03-24 | 2004-03-04 | Buenger Joachim | Use of ectoin or ectoin derivatives for protecting stress proteins in the skin |
US20030114324A1 (en) * | 2001-12-14 | 2003-06-19 | Rainer Lange | Cleansing compositions and their use in feminine hygiene wipes |
EP1407758A1 (de) * | 2002-10-10 | 2004-04-14 | Beiersdorf AG | Fettfreie Sonnenschutzmittel |
US20060029563A1 (en) * | 2002-12-30 | 2006-02-09 | Jean-Noel Thorel | Cutanceous metabolic bio-activator |
US20070155695A1 (en) * | 2004-01-19 | 2007-07-05 | Corinna Wirth | Flavonoid complexes with cyclodextrins |
US20070027223A1 (en) * | 2005-07-28 | 2007-02-01 | Werner Bruchert | Foamed preparation |
Non-Patent Citations (1)
Title |
---|
"INTERNATIONAL COSMETIC INGREDIENT DICTIONARY AND HANDBOOK, CTFA, 11th Ed", vol. 1, 1 January 2006, TARA E GOTTSCHALCK; GERALD N MCEWEN (EDITORS), WASHINGTON, D.C, pages: 560,1108, XP002580710 * |
Also Published As
Publication number | Publication date |
---|---|
US8293784B2 (en) | 2012-10-23 |
DE102007057543A1 (de) | 2009-06-04 |
US20110039924A1 (en) | 2011-02-17 |
JP2011504891A (ja) | 2011-02-17 |
EP2211827A2 (de) | 2010-08-04 |
WO2009068275A2 (de) | 2009-06-04 |
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